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The implications of target saturation for the use of drug–target residence time | Nature Reviews Drug Discovery
Covalent fragment libraries in drug discovery - ScienceDirect
Contribution of NIH funding to new drug approvals 2010–2016 | PNAS
DeepConv-DTI: Prediction of drug-target interactions via deep learning with convolution on protein sequences
Covalent fragment libraries in drug discovery - ScienceDirect
Biased Receptor Signaling in Drug Discovery | Pharmacological Reviews
Covalent fragment libraries in drug discovery - ScienceDirect
Drug development - Wikipedia
Creating and screening natural product libraries - Natural Product Reports (RSC Publishing) DOI:10.1039/C9NP00068B
Direct small-molecule inhibitors of KRAS: from structural insights to mechanism-based design | Nature Reviews Drug Discovery
Effects of target binding kinetics on in vivo drug efficacy: koff, kon and rebinding - Vauquelin - 2016 - British Journal of Pharmacology - Wiley Online Library
Biophysics in drug discovery: impact, challenges and opportunities | Nature Reviews Drug Discovery
Computational design of substrate selective inhibition
Macrocycles in new drug discovery | Future Medicinal Chemistry
Recent advances in combinatorial drug screening and synergy scoring - ScienceDirect
Screening-based approach to discover effective platinum-based chemotherapies for cancers with poor prognosis
CISNE: An accurate description of dose-effect and synergism in combination therapies | Scientific Reports
The drug–target residence time model: a 10-year retrospective | Nature Reviews Drug Discovery
Covalent fragment libraries in drug discovery - ScienceDirect
Organ‐on‐chip models: Implications in drug discovery and clinical applications - Mittal - 2019 - Journal of Cellular Physiology - Wiley Online Library
Development and optimization of a high-throughput screening method utilizing Ancylostoma ceylanicum egg hatching to identify novel anthelmintics
PDF) Theoretical Basis, Experimental Design, and Computerized Simulation of Synergism and Antagonism in Drug Combination Studies
Application of computational methods for anticancer drug discovery, design, and optimization - ScienceDirect
PDF) The nature of ligand efficiency
